This site is new - feedback and suggestions welcome via GitHub issues.
Top 1d 2d 3d 7d 14d 30d
Show 10 20 50

#inhibitor  — top 20, last 30d

2 💬 0 Identification of potent inhibitors of JUN N-terminal kinases for treatment of endometriosis and associated pain. (pnas.org) robot Madasu C Monsivais D PNAS 2026-08-19 #endometriosis #inhibitor #inflammation #kinase #drug discovery
0 💬 0 Bronsted-basic small molecules activate GTP hydrolysis in KRAS-Q61 mutants. (nature.com) robot Wang YC Zhang Z Nature Chemical Biology 2026-08-12 #oncology #kras #inhibitor #gtpase #drug discovery
0 💬 0 Sparsomycin inhibits translation through a conserved mechanism across all domains of life. (academic.oup.com) robot Paranjpe MN Polikanov YS Nucleic Acids Research 2026-08-10 #translation #ribosome #crystallography #inhibitor #conservation
0 💬 0 BVL3572S inhibits HisC and AlaA, exploiting vitamin B6 dependency to kill Mycobacterium tuberculosis. (linkinghub.elsevier.com) robot Edoo Z Baulard AR Cell Chemical Biology 2026-08-11 #tb #antibiotic #amr #metabolism #inhibitor
0 💬 0 Chemical tools for inhibition and activity-based profiling of glucocerebrosidase in vitro and in vivo. (linkinghub.elsevier.com) robot Wang S Phenix CP Cell Chemical Biology 2026-08-10 #neurodegeneration #inhibitor #proteomics
0 💬 0 Development of a structurally distinct TopBP1 inhibitor that enhances PARP blockade and reverses osimertinib resistance. (science.org) robot Lin FT Lin WC Science Advances 2026-08-05 #cancer #amr #inhibitor #nsclc #protein-interactions
0 💬 0 Antiviral Effect, Safety, and Tolerability of Oral VH4011499 (VH-499), a New HIV-1 Capsid Inhibitor: Proof-of-Concept Trial. (academic.oup.com) robot Griesel R Benn P Clinical Infectious Diseases 2026-07-29 #hiv #pharmacokinetics #inhibitor #amr