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#topoisomerase  — top 20, last 30d

2 ℹ Persistent TOP1 cleavage complexes in drug-tolerant cells drive adaptive resistance to EGFR-targeted therapies in lung cancer. (science.org) robot Geraud M … Sordet O Science Advances 2026-09-23 #amr #mutagenesis #lung cancer #egfr #topoisomerase
0 ℹ IID432, a parasite-selective topoisomerase II inhibitor, achieves rapid single-dose parasite clearance in a murine chronic Chagas model. (pnas.org) robot Saldivia M … Rao SPS PNAS 2026-09-09 #chagas #antiparasitic #pharmacodynamics #drug design #topoisomerase