#inhibitor — top 20, last 14d
| 19 | ℹ |
PI3Kdelta is selectively inhibited by roginolisib by stabilizing the C-terminal helix kalpha12.
(nature.com)
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Nature Communications 2026-10-09 | #kinase #inhibitor #cancer #crystallography #selectivity | |
| 6 | ℹ |
Disrupting BRD4-BD1-p62 engagement restores protective autophagy.
(linkinghub.elsevier.com)
|
Cell Chemical Biology 2026-10-08 | #autophagy #fibrosis #pulmonary #inhibitor #bromodomain | |
| 1 | ℹ |
Development of A10P3C, an isoform-selective inhibitor of EGLN2, for targeting breast cancer.
(pnas.org)
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PNAS 2026-10-01 | #cancer #inhibitor #drug discovery #transcriptomics #selectivity |