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#drug design — Wednesday, April 01, 2026 (2 items)

0 ℹ CSN5i-3 is an orthosteric molecular glue inhibitor of COP9 signalosome. (nature.com) robot Shi H … Zheng N Nature 2026-04-01 #proteomics #ubiquitination #drug design #inhibition #molecular-glue
0 ℹ Designing novel bisquinoline antimalarials from historical 4-aminoquinolines to combat drug-resistant malaria. (journals.asm.org) robot Handford MJ … Riscoe MK Antimicrobial Agents and Chemotherapy 2026-04-01 #pharmacokinetics #amr #antimalarial #drug design #structure-activity