#drug design — Wednesday, April 01, 2026 (2 items)
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CSN5i-3 is an orthosteric molecular glue inhibitor of COP9 signalosome.
(nature.com)
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Nature 2026-04-01 | #proteomics #ubiquitination #drug design #inhibition #molecular-glue | |
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Designing novel bisquinoline antimalarials from historical 4-aminoquinolines to combat drug-resistant malaria.
(journals.asm.org)
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Antimicrobial Agents and Chemotherapy 2026-04-01 | #pharmacokinetics #amr #antimalarial #drug design #structure-activity |